الأبحاث

بهاء الدين مصطفى عدلى الجندى

أستاذ مساعد

كلية العلوم كيمياء

Identification of Novel Mitochondrial Pyruvate Carrier Inhibitors by Homology Modeling and Pharmacophore-Based Virtual Screening

2022

البحث الكامل الملخص

Ligand-based design, synthesis, computational insights, and in vitro studies of novel N-(5-Nitrothiazol-2-yl)-carboxamido derivatives as potent inhibitors of SARS-CoV-2 main protease

2022

البحث الكامل الملخص

Structure-based design and synthesis of conformationally constrained derivatives of methyl-piperidinopyrazole (MPP) with estrogen receptor (ER) antagonist activity

2022

Identification of novel small molecule inhibitors against the NS3/4A protease of hepatitis C virus genotype 4a

Bentham Science 2019

Synthesis and Evaluation of Troponoids as a New Class of Antibiotics

American Chemical Society 2019

Development of novel liver X receptor modulators based on a 1, 2, 4-triazole scaffold

Elsevier 2019

Identification of 4-isopropyl–thiotropolone as a novel anti-microbial: regioselective synthesis, NMR characterization, and biological evaluation

Royal Society of Chemistry 2018

Recent Advances in the Medicinal Chemistry of Liver X Receptors

American Chemical Society 2018

P450 3A-Catalyzed O-Dealkylation of Lapatinib Induces Mitochondrial Stress and Activates Nrf2

American Chemical Society 2016

Stereoselective Synthesis, Structural and Spectroscopic Study of 4, 5, 11-Triazatricyclo [6.2. 1.0* 2, 6*] Undec-5-ene

Wiley 2015

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Computational Chemistry

Drug Discovery

Medicinal Chemistry

Natural Products

Nuclear Hormone Receptors

Nuclear Magnetic Resonance (NMR)

Organic Synthesis